IT1248486B - Agente terapeutico ad attivita' sul sistema nervoso centrale - Google Patents

Agente terapeutico ad attivita' sul sistema nervoso centrale

Info

Publication number
IT1248486B
IT1248486B IT02041890A IT2041890A IT1248486B IT 1248486 B IT1248486 B IT 1248486B IT 02041890 A IT02041890 A IT 02041890A IT 2041890 A IT2041890 A IT 2041890A IT 1248486 B IT1248486 B IT 1248486B
Authority
IT
Italy
Prior art keywords
therapeutic agent
nervous system
central nervous
agent activities
activities
Prior art date
Application number
IT02041890A
Other languages
English (en)
Italian (it)
Other versions
IT9020418A0 (en]
IT9020418A1 (it
Inventor
Roberto Pellicciari
Flavio Moroni
Original Assignee
Roberto Pellicciari
Flavio Moroni
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roberto Pellicciari, Flavio Moroni filed Critical Roberto Pellicciari
Publication of IT9020418A0 publication Critical patent/IT9020418A0/it
Priority to IT02041890A priority Critical patent/IT1248486B/it
Priority to BR919106500A priority patent/BR9106500A/pt
Priority to EP91909910A priority patent/EP0532545A1/en
Priority to AU78832/91A priority patent/AU7883291A/en
Priority to PCT/EP1991/000950 priority patent/WO1991017750A1/en
Priority to JP91509723A priority patent/JPH05507086A/ja
Priority to HU9203634A priority patent/HUT64695A/hu
Priority to CA002083507A priority patent/CA2083507A1/en
Publication of IT9020418A1 publication Critical patent/IT9020418A1/it
Priority to NO924472A priority patent/NO924472D0/no
Application granted granted Critical
Publication of IT1248486B publication Critical patent/IT1248486B/it

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/455Nicotinic acids, e.g. niacin; Derivatives thereof, e.g. esters, amides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Biomedical Technology (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
IT02041890A 1990-05-24 1990-05-24 Agente terapeutico ad attivita' sul sistema nervoso centrale IT1248486B (it)

Priority Applications (9)

Application Number Priority Date Filing Date Title
IT02041890A IT1248486B (it) 1990-05-24 1990-05-24 Agente terapeutico ad attivita' sul sistema nervoso centrale
PCT/EP1991/000950 WO1991017750A1 (en) 1990-05-24 1991-05-21 Nicotinylalanine as a therapeutic agent acting on the central nervous system
EP91909910A EP0532545A1 (en) 1990-05-24 1991-05-21 Nicotinylalanine as a therapeutic agent acting on the central nervous system
AU78832/91A AU7883291A (en) 1990-05-24 1991-05-21 Nicotinylalanine as a therapeutic agent acting on the central nervous system
BR919106500A BR9106500A (pt) 1990-05-24 1991-05-21 Nicotinilalanina como agente terapeutico atuando sobre o sistema nervoso central
JP91509723A JPH05507086A (ja) 1990-05-24 1991-05-21 中枢神経系に作用する治療剤としてのニコチニルアラニン
HU9203634A HUT64695A (en) 1990-05-24 1991-05-21 Method for production of preparations containing nicotinyl-alanine for the treatment of central nervous system (cns) diseares
CA002083507A CA2083507A1 (en) 1990-05-24 1991-05-21 Nicotinylalanine as a therapeutic agent acting on the central nervous system
NO924472A NO924472D0 (no) 1990-05-24 1992-11-20 Nikotinylalanin som terapeutisk middel med virkning paa sentralnervesystemet

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT02041890A IT1248486B (it) 1990-05-24 1990-05-24 Agente terapeutico ad attivita' sul sistema nervoso centrale

Publications (3)

Publication Number Publication Date
IT9020418A0 IT9020418A0 (en]) 1990-05-24
IT9020418A1 IT9020418A1 (it) 1991-11-24
IT1248486B true IT1248486B (it) 1995-01-19

Family

ID=11166634

Family Applications (1)

Application Number Title Priority Date Filing Date
IT02041890A IT1248486B (it) 1990-05-24 1990-05-24 Agente terapeutico ad attivita' sul sistema nervoso centrale

Country Status (8)

Country Link
EP (1) EP0532545A1 (en])
JP (1) JPH05507086A (en])
AU (1) AU7883291A (en])
BR (1) BR9106500A (en])
CA (1) CA2083507A1 (en])
HU (1) HUT64695A (en])
IT (1) IT1248486B (en])
WO (1) WO1991017750A1 (en])

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0684238A3 (en) * 1994-04-27 1997-01-15 Hoffmann La Roche Process for the preparation of dicarboxamides.
US5536867A (en) * 1994-04-27 1996-07-16 Hoffmann-La Roche Inc. Process for the manufacture of dicarboxamides
AU707084B2 (en) * 1995-03-14 1999-07-01 Edward G. Shaskan Compositions comprising nicotynylalanine and an inhibitor of glycine conjugation or vitamin B6
RU2742765C1 (ru) * 2017-09-28 2021-02-10 ЭлДжи КЕМ, ЛТД. Способ получения промежуточного соединения для синтеза лекарственного средства

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3649649A (en) * 1967-07-10 1972-03-14 Nisso Kako Co Ltd Fluoran derivatives and preparation thereof
FR1596106A (en]) * 1968-12-13 1970-06-15
US4065566A (en) * 1975-04-17 1977-12-27 Interx Research Corporation N-Nicotinoyl-3,4-dinicotinoyloxy-L-phenylalanine and derivatives pharmaceutical compositions and methods containing same

Also Published As

Publication number Publication date
BR9106500A (pt) 1993-05-25
HU9203634D0 (en) 1993-03-29
AU7883291A (en) 1991-12-10
JPH05507086A (ja) 1993-10-14
IT9020418A0 (en]) 1990-05-24
IT9020418A1 (it) 1991-11-24
CA2083507A1 (en) 1991-11-25
EP0532545A1 (en) 1993-03-24
HUT64695A (en) 1994-02-28
WO1991017750A1 (en) 1991-11-28

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Legal Events

Date Code Title Description
0001 Granted